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產品基本信息 |
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產品編號:122333 |
產品名稱:阿齊沙坦, ≥98% (HPLC) |
產品CAS:147403-03-0 |
規格含量:10mg |
產品價格:930 |
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產品詳細介紹 |
阿齊沙坦, ≥98% (HPLC)
Product Name: Azilsartan
CAS號: 147403-03-0
分子式: C25H20N4O5
分子量: 456.45
用途: 阿齊沙坦(又稱阿齊沙坦酯,英語:Azilsartan)(INN) 是一款正處于研發中的治療高血壓癥的血管緊張素II受體拮抗劑藥物,多用于治療高血壓癥,也是目前唯一處于末期臨床的血管緊張素II受體拮抗劑(沙坦類)藥物。
貯存:儲存溫度2-8°C
生化和生理學機理:Azilsartan is a highly potent and slowly dissociating Angiotensin II type 1 (AT1) receptor blocker (ARB) with an IC50 of 2.6 nM. It is the active form of Azilsartan medoxomil, used for treatment of hypertension. Azilsartan may also have potentially beneficial effects on metabolic syndrome including insulin sensitizing activity that may involve more than just blockade of AT(1) receptors.
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